Monday, April 2, 2012

Asgn_24B_Class_33_Article_21_2012_04_04

Read Article  21: Meindert Danhof, Joost de Jongh, Elizabeth C. M. De Lange, Oscar Della Pasqua, Bart A. Ploeger, and Rob A. Voskuyl. Mechanism-Based Pharmacokinetic-Pharmacodynamic Modeling: Biophase Distribution, Receptor Theory, and Dynamical Systems Analysis. Annu.Rev.Pharmacol.Toxicol. 47 (1):357-400, 2007. (RefID_20183). Get an overview of the content and be prepared to discuss each figure in detail. Post a PCRC.

3 comments:

  1. Brian Evans
    24B/Mech based PKPD modeling

    0. Knew: I was familiar with many of the mathematical models introduced in the text, from compartmental models to interactive pathways such as competition and allosterism.

    1. Learned: That PK/PD modeling is much more complicated and advanced than I was previously aware, and that more complex, synergistic models are now being created in a sort of systems biology approach to PK/PD modeling.

    2. Pressing ?: How can we account for the differences in PK/PD parameters between milli 1.0 and a full sized human?

    3. Presentation: Physiological counter-regulatory mechanisms

    4. Thoughts: This was a very thorough paper, I look forward to reading the text in entirety as opposed to skimming it. I like that the models and examples discussed were separated into mechanism based categories, it helped me understand the reasoning behind the math.

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  2. Will Matloff
    24B/Mechanism based PK/PD Modeling

    0. Knew: Basics of PK/PD modeling.

    1. Learned: Fundamentals of mechanism based PK/PD modeling. These models characterize the causal mechanisms between the administration of a drug and its response.

    2. Pressing?: Are there any specific characteristics of certain drugs that make them more effectively modeled by mechanism-based PDMD models?

    3. Presentation: The role of homeostatic mechanisms in PK/PD.

    4. Thoughts: It seems very natural to use mechanism based models. It is nice that with mechanism based modeling, organism-independent parameters can be found, which is useful for HoCs.

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  3. Zach Eagleton
    24B/Mechanism based PK/PD modeling
    0 Knew: Basics of Pk/PD modeling
    1 Learned: How mechanism based PK/PD modeling works. The multiple steps between administration and effect.
    2 Pressing ?: From a systems biology perspective how well do these models model the extreme patient cases?
    3 Presentation: Allosterism
    4 Thoughts: After skimming this article it looks very in-depth with sufficient math backing it up.

    ReplyDelete